Histone Acetyltransferase Inhibitor II 是一种选择性的细胞渗透性 p300 组蛋白乙酰转移酶抑制剂，IC50值为 5 μM。它在哺乳动物细胞中具有抗乙酰化酶活性，可用于癌症研究。

Histone Acetyltransferase Inhibitor II is a selective and cell permeable inhibitor of p300 histone acetyltransferase(IC50 : 5 μM).with anti-acetylase activity in mammalian cells.

Histone Acetyltransferase Inhibitor II (compound 2c) was the most active inhibitor, also showing high specificity for p300 as compared to other histone acetyltransferases.?Most notably, 2c showed anti-acetylase activity in mammalian cells.

932749-62-7

C20H16Br2O3

464.15

DMSO:30 mg/mL (64.63 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years