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GSK251
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
GSK251图片
CAS NO:2125968-05-8
包装与价格:
包装价格(元)
1mg电议
5mg电议
10mg电议

产品介绍
GSK251 是一种高效、高选择性、口服生物利用度的 PI3Kδ 抑制剂,具有新颖的结合模式。
Cas No.2125968-05-8
分子式C29H37FN6O4S
分子量584.71
溶解度DMSO : 62.5 mg/mL (106.89 mM; ultrasonic and warming and heat to 60℃)
储存条件Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

GSK251 is a highly potent, highly selective, orally bioavailable inhibitor of PI3Kδ with a novel binding mode.

[1]. Down K, et al. Discovery of GSK251: A Highly Potent, Highly Selective, Orally Bioavailable Inhibitor of PI3Kδ with a Novel Binding Mode. J Med Chem. 2021 Sep 23;64(18):13780-13792.