Catalog No. | Product Name | Summary | Targets | CAS Number | Smiles |
A3001 | PCI-32765 (Ibrutinib) | Bruton's tyrosine kinase (BTK) inhibitor | BTK | 936563-96-1 | C=CC(=O)N1CCCC(C1)N2C3=C(C(=N2)C4=CC=C(C=C4)OC5=CC=CC=C5)C(=NC=N3)N |
A3302 | CGI-1746 | Btk inhibitor | BTK | 910232-84-7 | CC1=C(C=CC=C1NC(=O)C2=CC=C(C=C2)C(C)(C)C)C3=CN(C(=O)C(=N3)NC4=CC=C(C=C4)C(=O)N5CCOCC5)C |
A4506 | DMOG | Competitive HIF-PH inhibitor, cell-permeable | HIF | 89464-63-1 | COC(=O)CNC(=O)C(=O)OC |
A8164 | Cyclo (-RGDfK) | Inhibitor of αvβ3 integrin | Integrin | 161552-03-0 | C1C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)N1)CCCN=C(N)N)CCCCN)CC2=CC=CC=C2)CC(=O)O |
A8233 | DMXAA (Vadimezan) | Tumnor vascular disrupting agent, apoptosis inducer | VDA | 117570-53-3 | CC1=C(C2=C(C=C1)C(=O)C3=C(O2)C(=CC=C3)CC(=O)O)C |
A8660 | Cilengitide | Integrin inhibitor for αvβ3 and αvβ5 | Integrin | 188968-51-6 | CC(C)C1C(=O)NC(C(=O)NCC(=O)NC(C(=O)NC(C(=O)N1C)CC2=CC=CC=C2)CC(=O)O)CCCN=C(N)N |
B3708 | RGD (Arg-Gly-Asp) Peptides | Inhibits integrin binding to RGD motifs | Integrin | 99896-85-2 | C(CC(C(=O)NCC(=O)NC(CC(=O)O)C(=O)O)N)CN=C(N)N |
B6004 | PX-478 2HCl | HIF-1α inhibitor | HIF | 685898-44-6 | ClCC[N+](C1=CC=C(C[C@@](N)([H])C(O)=O)C=C1)([O-])CCCl.Cl.Cl |