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Umbralisib R-enantiomer
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Umbralisib R-enantiomer图片
CAS NO:1532533-69-9
包装与价格:
包装价格(元)
2mg电议
5mg电议
10mg电议
50mg电议

产品名称
TGR-1202 R-enantiomer
RP5264 R-enantiomer
产品介绍
Umbralisib R-enantiomer (TGR-1202 R-enantiomer) 是PI3Kδ抑制剂,是 TGR-1202 活性较低的对映体。
生物活性

Umbralisib R-enantiomer (TGR-1202 R-enantiomer) is aPI3Kδinhibitor, which is the less active enantiomer of TGR-1202.

IC50& Target[1]

PI3Kδ

 

体外研究
(In Vitro)

Umbralisib R-enantiomer (TGR-1202 R-enantiomer) (Formula A) exhibits a 50% inhibitory concentration (IC50) with respect to the δ type PI3-kinase that is at least 20-fold lower than the inhibitor's IC50with respect to the rest of the other PI3K isoforms (i.e., a, β, and γ)[1].

分子量

571.55

性状

Solid

Formula

C31H24F3N5O3

CAS 号

1532533-69-9

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式
Powder-20°C3 years
4°C2 years
In solvent-80°C6 months
-20°C1 month