CAS NO: | 1532533-69-9 |
包装 | 价格(元) |
2mg | 电议 |
5mg | 电议 |
10mg | 电议 |
50mg | 电议 |
生物活性 | Umbralisib R-enantiomer (TGR-1202 R-enantiomer) is aPI3Kδinhibitor, which is the less active enantiomer of TGR-1202. | ||||||||||||
IC50& Target[1] |
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体外研究 (In Vitro) | Umbralisib R-enantiomer (TGR-1202 R-enantiomer) (Formula A) exhibits a 50% inhibitory concentration (IC50) with respect to the δ type PI3-kinase that is at least 20-fold lower than the inhibitor's IC50with respect to the rest of the other PI3K isoforms (i.e., a, β, and γ)[1]. | ||||||||||||
分子量 | 571.55 | ||||||||||||
性状 | Solid | ||||||||||||
Formula | C31H24F3N5O3 | ||||||||||||
CAS 号 | 1532533-69-9 | ||||||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||||||
储存方式 |
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