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E4CPG
本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。
E4CPG图片
CAS NO:170846-89-6
包装与价格：
包装价格(元)
10mg电议
50mg电议

产品介绍
E4CPG ((RS)-ECPG) 是 I 组/II 组代谢型谷氨酸受体 (mGluR) 拮抗剂。
Cas No.170846-89-6
别名(RS)-ECPG
化学名(S)-4-(1-amino-1-carboxypropyl)benzoic acid
Canonical SMILESOC([C@](CC)(C1=CC=C(C(O)=O)C=C1)N)=O
分子式C11H13NO4
分子量223.23
溶解度Soluble to 100 mM in 1.1eq. NaOH
储存条件Store at RT
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

E4CPG is a novel group I/group II metabotropic glutamate receptor antagonist, more potent than (RS)-MCPG .

References:
[1]. Sekiyama N et al. Structure-activity relationships of new agonists and antagonists of different metabotropic glutamate receptorsubtypes. Br J Pharmacol, 1996 Apr, 117(7):1493-503.
[2]. Bedingfield JS et al. Structure-activity relationships for a series of phenylglycine derivatives acting at metabotropic glutamate receptors (mGluRs). Br J Pharmacol. 1995 Dec;116(8):3323-9.