Metergoline 是一种血清素 (5-HT) 受体和多巴胺受体拮抗剂，对 5-HT2A、5-HT2B 和 5-HT2C 的 pKis 分别为 8.64、8.75 和 8.75。
| Cas No. | 17692-51-2 |
| 别名 | 甲麦角林 |
| 化学名 | benzyl (((6aR,9S,10aR)-4,7-dimethyl-4,6,6a,7,8,9,10,10a-octahydroindolo[4,3-fg]quinolin-9-yl)methyl)carbamate |
| Canonical SMILES | O=C(NC[C@@H]1C[C@H]2[C@@H](CC3=CN(C)C4=CC=CC2=C34)N(C)C1)OCC5=CC=CC=C5 |
| 分子式 | C25H29N3O2 |
| 分子量 | 403.52 |
| 溶解度 | DMF: 30 mg/ml,DMF:PBS(pH7.2) (1:2): 0.3 mg/ml,DMSO: 25 mg/ml,Ethanol: 5 mg/ml |
| 储存条件 | Store at RT |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
| 产品描述 | Metergoline is a psychoactive drug of the ergoline chemical class which acts as a ligand for various serotonin and dopamine receptors. |
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