CAS NO: | 129693-13-6 |
包装 | 价格(元) |
100mg | 电议 |
250mg | 电议 |
500mg | 电议 |
生物活性 | Sp-8-CPT-cAMPS, a cAMP analog, is a potent and selective activator of the cAMP-dependentprotein kinas A (PKA I andPKAII). Sp-8-CPT-cAMPS selects site A of RI compares to site A of RII by 153-fold and site B of RII compares to site B of RI by 59-fold[1][2]. |
IC50& Target | PKA[1] |
体外研究 (In Vitro) | Sp-8-CPT-cAMPS (100 μM; 24 h) enhances the IL-1β-stimulated nitrite release, and increases the release ofnitrite by vascular smooth muscle cells by 3 fold in the absence of IL-1β in vascular smooth muscle cells[2]. |
分子量 | 487.88 |
Formula | C16H15ClN5O5PS2 |
CAS 号 | 129693-13-6 |
运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |