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Letrozole-d4
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Letrozole-d4图片
CAS NO:1133712-96-5
包装与价格:
包装价格(元)
1mg电议
10mg电议

产品名称
来曲唑 d4
产品介绍
Letrozole-d4 是 Letrozole 的氘代物。Letrozole (CGS 20267) 是一种有效的,选择性的,可逆的和具有口服活性的非甾体类芳香化酶 (aromatase) 抑制剂,IC50值为 11.5 nM。Letrozole 选择性抑制雌激素的生物合成,可用于乳腺癌的研究。
生物活性

Letrozole-d4 (CGS 20267-d4) is the deuterium labeled Letrozole. Letrozole (CGS 20267) is a potent, selective, reversible and orally active non-steroidal inhibitor ofaromatase, with anIC50of 11.5 nM. Letrozole selective inhibits estrogen biosynthesis, and can be used for the research of breastcancer[1][2][3].

体外研究
(In Vitro)

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].

分子量

289.33

Formula

C17H7D4N5

CAS 号

1133712-96-5

中文名称

来曲唑 d4

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.