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AGN 193109-d7
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
AGN 193109-d7图片
CAS NO:1216429-25-2
包装与价格:
包装价格(元)
1mg电议
10mg电议

产品介绍
AGN 193109-d7 是 AGN 193109 的氘代物。AGN 193109 是一种视黄酸类似物,是有效的,特异性的视黄酸受体 (RARs) 拮抗剂,可抑制RARαRARβRARγ的活性,Kd值分别为 2 nM,2 nM 和 3 nM。
生物活性

AGN 193109-d7 is the deuterium labeled AGN 193109. AGN 193109 is a retinoid analog, and acts as a specific and highly effective antagonist ofretinoic acid receptors (RARs), withKds of 2 nM, 2 nM, and 3 nM forRARα,RARβ, andRARγ, respectively.

体外研究
(In Vitro)

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].

分子量

399.53

Formula

C28H17D7O2

CAS 号

1216429-25-2

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.