GR 94800 是一种有效的选择性 NK2 受体肽拮抗剂，对 NK2、NK1 和 NK3 受体的 pKB 值分别为 9.6、6.4 和 6.0。
| Cas No. | 141636-65-9 |
| 化学名 | (S)-1-((R)-1-((3S,6S,9R,12S)-9-((1H-indol-3-yl)methyl)-12-benzyl-3,6-dimethyl-1,4,7,10-tetraoxo-1-phenyl-2,5,8,11-tetraazatridecan-13-oyl)pyrrolidine-2-carbonyl)-N-((S)-1-amino-1-oxohexan-2-yl)pyrrolidine-2-carboxamide |
| Canonical SMILES | O=C([C@@H]1N(C([C@H](CC2=CC=CC=C2)NC([C@@H](CC3=CNC4=CC=CC=C34)NC([C@H](C)NC([C@H](C)NC(C5=CC=CC=C5)=O)=O)=O)=O)=O)CCC1)N6[C@H](C(N[C@H](C(N)=O)CCCC)=O)CCC6 |
| 分子式 | C49H61N9O8 |
| 分子量 | 904.08 |
| 溶解度 | Soluble to 4 mg/ml in ethanol |
| 储存条件 | Desiccate at -20°C |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
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