UFP-101 是一种有效的、选择性的、竞争性的 NOP 受体拮抗剂,pKi 为 10.24。
Cas No. | 849024-68-6 |
别名 | 竞争性沉默拮抗剂UFP-101 |
化学名 | (S,Z)-6-amino-N-((S,Z)-1-(((S)-6-amino-1-hydroxy-1-iminohexan-2-yl)imino)-5-guanidino-1-hydroxypentan-2-yl)-2-((Z)-((4Z,7Z,10Z,12S,13Z,15S,16Z,19Z,21S,22Z,24S,25Z,27S,28Z,30S,31Z,33S,34Z,36S)-27-(4-aminobutyl)-12-benzyl-24,36-bis(3-guanidinopropyl)-4,7,10 |
Canonical SMILES | C[C@@](/N=C(O)/C/N=C(O)/[C@](/N=C(O)/[C@](/N=C(O)/C/N=C(O)/C/N=C(O)/CNCC1=CC=CC=C1)([H])CC2=CC=CC=C2)([H])[C@@](O)([H])C)([H])/C(O)=N/[C@@](/C(O)=N/[C@@](/C(O)=N/[C@@](/C(O)=N/[C@@](/C(O)=N/[C@@](/C(O)=N/[C@@](/C(O)=N/[C@@](/C(O)=N/[C@@](C(O)=N)([H])CCCCN |
分子式 | C82H138N32O21 |
分子量 | 1665.94 |
溶解度 | Soluble to 1 mg/ml in Water |
储存条件 | Desiccate at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |