ISAM-140 (22b) 是一种有效的、高选择性的A2Badenosine receptor拮抗剂,其Ki值为 3.49 nM。
生物活性 | ISAM-140 (22b) is a potent and highly selectiveA2Badenosine receptorantagonist with aKiof 3.49 nM[1]. |
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体外研究 (In Vitro) | ISAM-140 (22b) (0.1-100 μM) inhibits NECA (5'-N-ethylcarboxamido adenosine)-stimulated cAMP accumulation[1]. ISAM-140 shows a KBvalue of 27.00 nM[1].
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |