CAS NO: | 180304-07-8 |
包装 | 价格(元) |
5mg | 电议 |
10mg | 电议 |
生物活性 | S-22153 is a potentmelatonin receptorantagonist withEC50values of 19 nM, 4.6 nM forhMT1andhMT2melatonin receptor, respectively. S-22153 hasKivalues of 8.6 nM (CHO cells) and 16.3 nM (HEK cells) for hMT1, and 6.0 nM (CHO cells) and 8.2 nM (HEK cells) for hMT2. S-22153 is a specific ligand of MT1and MT2melatonin receptors subtypes[1][2]. | ||||||||
IC50& Target[2] |
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体内研究 (In Vivo) | S-22153 sets the temperature and activity periods to approximately 24 hr and increase the circadian amplitude of both rhythms in mice, which exposed to continuous light[1].
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分子量 | 247.36 | ||||||||
Formula | C14H17NOS | ||||||||
CAS 号 | 180304-07-8 | ||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |