CAS NO: | 146669-29-6 |
包装 | 价格(元) |
10 mM * 1 mL in DMSO | 电议 |
5mg | 电议 |
10mg | 电议 |
25mg | 电议 |
50mg | 电议 |
100mg | 电议 |
200mg | 电议 |
500mg | 电议 |
生物活性 | (RS)-MCPG (alpha-MCPG) is a competitive and selective group I/group IImetabotropic glutamate receptor (mGluR)antagonist. (RS)-MCPG blocks theta-burst stimulation (TBS)-induced shifts in both juvenile and neonatal rat hippocampal neurons[1][2]. | ||||||||||||||||
IC50& Target | group I/group II mGluR[1] | ||||||||||||||||
体外研究 (In Vitro) | MCPG can block group I (mGluR1 and mGluR5) and group II receptors (mGluR2 and mGluR3)[2]. | ||||||||||||||||
体内研究 (In Vivo) | (RS)-MCPG (alpha-MCPG; 500 μM) blocks the TBS-induced shifts in EGABA in either juvenile or neonatal neurons[1]. | ||||||||||||||||
分子量 | 209.20 | ||||||||||||||||
性状 | Solid | ||||||||||||||||
Formula | C10H11NO4 | ||||||||||||||||
CAS 号 | 146669-29-6 | ||||||||||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||||||||||
储存方式 |
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溶解性数据 | In Vitro: 1M NaOH : 100 mg/mL(478.01 mM;ultrasonic and adjust pH to 10 with NaOH) DMSO : 6 mg/mL(28.68 mM;Need ultrasonic and warming) H2O :< 0.1 mg/mL (ultrasonic;heat to 80℃)(insoluble) 配制储备液
* 请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。 |