CAS NO: | 1276617-62-9 |
包装 | 价格(元) |
100mg | 电议 |
250mg | 电议 |
500mg | 电议 |
生物活性 | VU0409106 is a potent and selectivemGlu5negative allosteric modulator (NAM) with anIC50of 24 nM. VU0409106 shows anxiolytic effects in rat models in a concentration-dependent manner. VU0409106 also penetrates the blood-brain barrier (BBB)[1][2]. | ||||||||||||||||||||||||
IC50& Target |
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体内研究 (In Vivo) | VU0409106 (10 mg/kg; i.p.; once) penetrates the blood-brain barrier (BBB) and demonstrates good brain to plasma ratio that near unity[1].
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分子量 | 330.34 | ||||||||||||||||||||||||
Formula | C15H11FN4O2S | ||||||||||||||||||||||||
CAS 号 | 1276617-62-9 | ||||||||||||||||||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||||||||||||||||||
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |