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MRS2365
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
MRS2365图片
CAS NO:436847-09-5
包装与价格:
包装价格(元)
100mg电议
250mg电议
500mg电议

产品介绍
MRS2365 是一种有效的选择性P2Y1受体激动剂,EC50为 0.4 nM。MRS2365 对 P2Y12 或 P2Y13 受体几乎没有激动或拮抗活性。
生物活性

MRS2365 is a potent and selectiveP2Y1 receptoragonist with anEC50of 0.4 nM. MRS2365 shows little agonist or antagonist activity at the P2Y12 or P2Y13 receptors[1][2].

体外研究
(In Vitro)

Selective activation of the P2Y1 receptor also is suggested from functional studies of human platelets as MRS2365 potently induced shape change without causing the sustained aggregation that is a hallmark of simultaneous activation of the P2Y1 and P2Y12 receptors by ADP or by previously studied ADP analogues[2].

分子量

483.33

Formula

C13H19N5O9P2S

CAS 号

436847-09-5

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.