CAS NO: | 252845-37-7 |
包装 | 价格(元) |
100mg | 电议 |
250mg | 电议 |
500mg | 电议 |
生物活性 | Veldoreotide (DG3173) a somatostatin analogue, that can bind to and activate thesomatostatin receptors (SSTR) 2, 4, and 5. Veldoreotide inhibitsgrowth hormone (GH)secretion in adenomas compared withOctreotide(HY-P0036). Veldoreotide has the potential to be used as pain modulating agent[1] | ||||||||
IC50& Target[1] |
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体外研究 (In Vitro) | Veldoreotide stimulates the SST2, SST4, and SST5 receptors with high potency and efficacy in the HEK293 cells, co-expressing these receptors with the GIRK2 channels; EC50s of 37.6 ± 4.5 nM, 31.3 ± 14.4 nM and 10.5 ± 3.4 nM for GIRK2-SST2, GIRK2-SST4 and GIRK2-SST5, respectively[1]. Cell Proliferation Assay[1]
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Clinical Trial | |||||||||
分子量 | 1123.30 | ||||||||
Formula | C60H74N12O10 | ||||||||
CAS 号 | 252845-37-7 | ||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |