包装 | 价格(元) |
100mg | 电议 |
250mg | 电议 |
500mg | 电议 |
生物活性 | d[Cha4]-AVP TFA is a potent and selectivevasopressin (AVP) V1b receptoragonist with aKiof 1.2 nM forhuman V1b receptor. d[Cha4]-AVP TFA shows more selective for V1b receptor than human V1a receptor, V2 receptor, and oxytocin receptors[1][2]. |
IC50& Target | Ki: 1.2 nM (vasopressin V1B receptor), 151 nM (vasopressin V1A receptor), 240 nM (Oxytocin receptor), 750 nM (vasopressin V2 receptor) |
体外研究 (In Vitro) | d[Cha4]-AVP binds to hV1b receptors and human oxytocin receptors with pKivalues of 9.68 and 7.68, respectively[2]. |
分子量 | 1208.33 |
Formula | C52H72F3N13O13S2 |
Sequence | {Mpa}-Tyr-Phe-{Cha}-Asn-Cys-Pro-Arg-Gly-NH2 (Disulfide bridge:Mpa1-Cys6) |
Sequence Shortening | {Mpa}YF{Cha}NCPRG-NH2 (Disulfide bridge:Mpa1-Cys6) |
运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |