Rivaroxaban D4 (BAY 59-7939 D4) 是 Rivaroxaban 的氘代物。Rivaroxaban 是一种高效,选择性凝血因子 Xa (FXa) 抑制剂,IC50为 0.7 nM,Ki为 0.4 nM。
生物活性 | Rivaroxaban D4 (BAY 59-7939 D4) is a deuterium labeled Rivaroxaban. Rivaroxaban is a highly potent,selective and directFactor Xa(FXa) inhibitor, achieving a strong gain in anti-FXa potency (IC500.7 nM;Ki0.4 nM)[1][2]. |
IC50& Target | IC50: 0.7 nM (Factor Xa); Ki: 0.4 nM (Factor Xa)[1][2] |
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Powder | -20°C | 3 years | | 4°C | 2 years | In solvent | -80°C | 6 months | | -20°C | 1 month |
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