TM5007 是具有口服活性的纤溶酶原激活物抑制剂-1 (PAI-1) 的一种有效抑制剂,其IC50值为 29 μM,可增强纤溶活性并抑制凝血。TM5007 还能防止博莱霉素引起的小鼠肺纤维化过程。
生物活性 | TM5007 is a poent and orally active inhibitor of plasminogen activator inhibitor-1 (PAI-1) with anIC50of 29 μM. TM5007 enhance fibrinolysis activity and inhibits coagulation. TM5007 also prevents the fibrotic process initiated by bleomycin in mouse lung[1]. |
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |