Cimoxatone

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Cimoxatone

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:

73815-11-9

包装与价格：

包装	价格(元)
100mg	电议
250mg	电议
500mg	电议

产品名称

MD 780515

产品介绍

Cimoxatone (MD 780515) 是一种可逆的口服活性 A 型单胺氧化酶 (MAO-A) (type A monoamine oxidase (MAO-A)) 抑制剂。Cimoxatone 增强type A monoamine oxidase (MAO-A)的厌食作用。

生物活性

Cimoxatone (MD 780515) is a reversible, selectively and orally activetype Amonoamine oxidase(MAO-A)inhibitor. Cimoxatone enhances the anorectic action ofSerotonin(HY-B1473A)^[1].

IC₅₀& Target^[1]

MAO-A

体内研究
(In Vivo)

Cimoxatone (20 mg/kg; p.o.) 增强 5-HT (1 mg/kg; s.c.) 对大鼠的厌食作用^[1]。

Animal Model:	250-300 g, Adult male Wistar rats^[1]
Dosage:	20 mg/kg
Administration:	P.o.
Result:	Significiantly reduced sucrose intake induced by 1 mg/kg 5-HT or its vehicle injected 2 and 24 h later, significantly enhanced the anorectic action of 5-HT at 2 h but not at 24 h.

分子量

338.36

Formula

C₁₉H₁₈N₂O₄

CAS 号

73815-11-9

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.