Isamoltane hemifumarate 是 5-HT1B 受体的选择性拮抗剂，抑制 [125I]ICYP 与大鼠脑膜中 5-HT1B 识别位点的结合，IC50 为 39 nM。
| Cas No. | 874882-92-5 |
| 化学名 | 1-(2-(1H-pyrrol-1-yl)phenoxy)-3-(isopropylamino)propan-2-ol hemifumarate |
| Canonical SMILES | CC(NCC(O)COC1=CC=CC=C1N2C=CC=C2)C.CC(NCC(O)COC3=CC=CC=C3N4C=CC=C4)C.O=C(O)/C([H])=C([H])/C(O)=O |
| 分子式 | C16H22N2O2.½C4H4O4 |
| 分子量 | 332.4 |
| 溶解度 | <3.32mg/ml in Water |
| 储存条件 | Store at -20℃ |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
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