包装 | 价格(元) |
100mg | 电议 |
250mg | 电议 |
500mg | 电议 |
生物活性 | CBP/p300-IN-20 is a potent and selectivep300/CBPinhibitor, with apIC50of 10.1 for p300. CBP/p300-IN-20 can be used for the research ofcancer[1]. | ||||||||
IC50& Target[1] |
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体外研究 (In Vitro) | CBP/p300-IN-20 (compound 28) decreases Myc protein in cell-based cMyc HTRF assay, with a pEC50of 8.5[1]. Western Blot Analysis[1]
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体内研究 (In Vivo) | CBP/p300-IN-20 (compound 28) (0.54 mg/kg; i.v.) exhibits Cmax(210 ng/mL), AUC0→∞(102 hong/mL), CL (95 mL/min/kg), and T1/2(0.3 h) in rats[1]. | ||||||||
分子量 | 477.87 | ||||||||
Formula | C22H19ClF3N5O2 | ||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |