P300 bromodomain-IN-1 (Compoun 1u) 是一种有效的p300 (EP300) bromodomain抑制剂,IC50值为 49 nM。P300 bromodomain-IN-1 抑制c-Myc的表达,诱导 OPM-2 细胞 G1/G0 期阻滞和凋亡 (apoptosis)。
生物活性 | P300 bromodomain-IN-1 (Compoun 1u) is a potentp300 (EP300) bromodomaininhibitor with anIC50of 49 nM. P300 bromodomain-IN-1 suppresses the expression ofc-Mycand induces G1/G0 phase arrest andapoptosisin OPM-2 cells[1]. |
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |