您好,欢迎来到化工原料网! [登录] [免费注册]
化工原料网
位置:首页 > 产品库 > Etifoxine-d5
立即咨询
咨询类型:
     
*姓名:
*电话:
*单位:
Email:
*留言内容:
请详细说明您的需求。
*验证码:
 
Etifoxine-d5
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Etifoxine-d5图片
CAS NO:1346598-10-4
包装与价格:
包装价格(元)
100mg电议
250mg电议
500mg电议

产品介绍
Etifoxine-d5 是 Etifoxine 的氘代物。Etifoxine 是一个非苯二氮卓类的、具有 GABA 能的化合物,是GABAA受体亚基 α1β2γ2 和 α1β3γ2 的阳性变构调节剂。Etifoxine 在啮齿类动物中显示出抗焦虑和抗惊厥活性。
生物活性

Etifoxine-d5 is the deuterium labeled Etifoxine. Etifoxine, a non-benzodiazepine GABAergic compound, is a positive allosteric modulator of α1β2γ2 and α1β3γ2 subunit-containingGABAAreceptors. Etifoxine reveals anxiolytic and anticonvulsant properties in rodents[1][2][3].

体外研究
(In Vitro)

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].

分子量

305.81

Formula

C17H12D5ClN2O

CAS 号

1346598-10-4

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.