Raloxifene 6-Monomethyl Ether (Compound 7) is a Raloxifene derivative that inhibitsestrogen receptorα. Raloxifene 4-Monomethyl Ether inhibits MCF-7 cells with anIC₅₀of 250 nM and apIC₅₀of 6.6^[1].

Raloxifene 6-Monomethyl Ether (Compound 7) is a Raloxifene derivative with a methoxy group on C6. Raloxifene 6-Monomethyl Ether holds poor ICsub>50value because of disruption to the hydrogen bond network and steric disfavor^[1].

487.61

C₂₉H₂₉NO₄S

178451-13-3

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