CAS NO: | 80751-65-1 |
包装 | 价格(元) |
100mg | 电议 |
250mg | 电议 |
500mg | 电议 |
生物活性 | SKF-82958 ((±)-SKF 82958) is adopamine D1 receptorfull agonist (K0.5=4 nM), displays selective for D1 over D2 receptors (K0.5=73 nM). SKF-82958 induces dopamine D1 receptor-dependentadenylate cyclaseactivity in rat striatal membranes (EC50=491 nM)[1]. | ||||||||
体内研究 (In Vivo) | SKF-82958 ((±)-SKF 82958) (0.003-0.1 mg/kg; i.p.) results in dose-dependent increases in responding on the SKF-82958 appropriate lever, with full substitution following administration of the SKF-82958 training dose 0.03 mg/kg. Increasing the dose of SKF-82958 also results in a significant reduction in response rate[2].
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分子量 | 329.82 | ||||||||
Formula | C19H20ClNO2 | ||||||||
CAS 号 | 80751-65-1 | ||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |