CAS NO: | 1432063-88-1 |
包装: | 1mg |
市场价: | 11500元 |
生物活性 | Sitagliptin-d4 (MK-0431-d4) phosphate is the deuterium labeled Sitagliptin phosphate. Sitagliptin phosphate (MK-0431 phosphate) is a potent inhibitor ofDPP4with anIC50of 19 nM in Caco-2 cell extracts[1][2]. |
体外研究 (In Vitro) | Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1]. |
分子量 | 509.33 |
Formula | C16H14D4F6N5O5P |
CAS 号 | 1432063-88-1 |
中文名称 | 磷酸西他列汀 d4 (磷酸盐) |
运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |