S1427 是一种反苯环丙胺衍生的LSD1抑制剂，IC50为 390 nM，Ki为 80 nM。S1427 抑制 hERG 通道，且具有微粒体稳定性。抑制 LSD1 可减少癌细胞的增殖。
| 生物活性 | S1427 is a tranylcypromine-derivedLSD1inhibitor with theIC50of 390 nM andKiof 80 nM. S1427 exhibits desirable hERG channel inhibition and microsomal stability profiles. Inhibition of LSD1 partially reduces the proliferation ofcancercells[1]. |
| IC50& Target | |
| 分子量 | |
| Formula | |
| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
m.cnreagent.com
