包装 | 价格(元) |
100mg | 电议 |
250mg | 电议 |
500mg | 电议 |
生物活性 | D4R antagonist-2 is a potent and selectiveD4Rantagonist with anIC50of 6.52 μM. D4R antagonist-2 displays very favorable in vitro PK parameters and has good brain penetration. D4R antagonist-2 has the potential for the research of Parkinson’s disease[1]. | ||||||||||||||||||||
IC50& Target |
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体外研究 (In Vitro) | D4R antagonist-2 (compound 11a) shows good activity with an Kiof 299.4 nM[1]. | ||||||||||||||||||||
体内研究 (In Vivo) | D4R antagonist-2 displays very favorable in vitro PK parameters and is brain pentrent (Kp=2.9)[1].
b>Pharmacokinetic Parameters of D4R antagonist-2 in rats[1].
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分子量 | 408.87 | ||||||||||||||||||||
Formula | C21H23ClF2N2O2 | ||||||||||||||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||||||||||||||
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |