Orexin receptor antagonist 4 是一种有效的选择性食欲素 2 受体 (OX2R) 拮抗剂，IC50为 4.27 nM。Orexin receptor antagonist 4 对 OX2R 的选择性是对 OX1R 的 61 倍 (IC50为 295 nM) (WO2018206959A1; example 1)。
| 生物活性 | Orexin receptorantagonist 4 is potent and selectiveorexin 2 receptor (OX2R)antagonist with anIC50of 4.27 nM.Orexin receptorantagonist 4 is 61-fold selective for the OX2R over the OX1R (IC50of 295 nM) (WO2018206959A1; example 1)[1]. |
| IC50& Target[1] | OX2Receptor 4.27 nM (IC50) | OX1Receptor 295 nM (IC50) |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
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