Sumatriptan succinate (GR 43175) 是一种具有口服活性的 5-HT1 受体激动剂，对 5-HT1D、5-HT1B 和 5-HT1A 受体的 Kis 值分别为 17 nM、27 nM 和 100 nM。
| Cas No. | 103628-48-4 |
| 别名 | 舒马普坦琥珀酸盐; GR 43175 |
| 化学名 | butanedioic acid;1-[3-[2-(dimethylamino)ethyl]-1H-indol-5-yl]-N-methylmethanesulfonamide |
| Canonical SMILES | CNS(=O)(=O)CC1=CC2=C(C=C1)NC=C2CCN(C)C.C(CC(=O)O)C(=O)O |
| 分子式 | C14H21N3O2S.C4H6O4 |
| 分子量 | 413.49 |
| 溶解度 | ≥ 136.8mg/mL in DMSO, ≥ 47.2 mg/mL in Water |
| 储存条件 | Store at 2-8℃ |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
| 产品描述 | Sumatriptan succinate is a selective 5-HT1 receptor agonist with specificity towards 5-HT1D, 5-HT1B and 5-HT1A. In addition, the physicochemical properties of Sumatriptan succinate can be characterized using FT-IR, HPLC, SEM and XRD. It has been reported |
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