Ipsapirone 是 5-HT1A 受体的部分激动剂,在高剂量时对 5-HT2 和 α1-肾上腺素能功能产生抑制作用。
产品描述
Ipsapirone is a partial agonist of 5-HT1A receptor and produces an inhibitory effect on 5-HT2 and the α1-adrenergic function at high doses.
体内活性
Ipsapirone (2.5-80 mg/kg) induces a mild hind limb abduction and a slight flattening of body posture at the highest dose. Ipsapirone (35 mg/kg; i.p.) decreases the body temperature in rats and mice.
Cas No.
95847-70-4
分子式
C19H23N5O3S
分子量
401.48
储存和溶解度
DMSO:Soluble
Powder: -20°C for 3 years
In solvent: -80°C for 2 years