您好,欢迎来到化工原料网! [登录] [免费注册]
化工原料网
位置:首页 > 产品库 > SCD1 inhibitor-3
立即咨询
咨询类型:
     
*姓名:
*电话:
*单位:
Email:
*留言内容:
请详细说明您的需求。
*验证码:
 
SCD1 inhibitor-3
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
SCD1 inhibitor-3图片
CAS NO:1282606-48-7
包装与价格:
包装价格(元)
1 mg电议
5 mg电议
10 mg电议
25 mg电议
50 mg电议
100 mg电议

产品名称
SCD1 inhibitor 17a
SCD1-IN-3
产品介绍
SCD1 inhibitor-3 是一种安全、有效的、具有口服活性的 SCD1 抑制剂。SCD1 inhibitor-3 可用于肥胖症、二型糖尿病、血脂异常等代谢性疾病,以及皮肤病、痤疮、癌症等的研究。

产品描述

SCD1 inhibitor-3 is a safe, potent and orally active SCD1 inhibitor. SCD1 inhibitor-3 can be used for the research of metabolic diseases such as obesity, type II diabetes and dyslipidemia, as well as skin diseases, acne and cancer.

体内活性

SCD1 inhibitor-3 (compound 17a) (5 mg/kg; p.o.; 4 hours) reduces the plasma C16:1/C16:0 triglycerides desaturation index by 54 % [1] . SCD1 inhibitor-3 (2~10 mg/kg; p.o.; 4 hours) makes a dose-responsive reduction of plasma triglycerides desaturation index [1] . Animal Model: Lewis rats [1] Dosage: 5 mg/kg Administration: P.o.; 4 hours Result: Reduced the plasma C16:1/C16:0 triglycerides desaturation index by 54 %. Animal Model: Lewis rats [1] Dosage: 2~10 mg/kg Administration: P.o.; 4 hours Result: A dose-responsive reduction of plasma triglycerides desaturation index[1].

Cas No.

1282606-48-7

分子式

C19H16FN7O2

分子量

393.37

别名

SCD1 inhibitor 17a;SCD1-IN-3

储存和溶解度

DMSO:35 mg/mL (89 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years