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CGP71683 hydrochloride
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
CGP71683 hydrochloride图片
CAS NO:192322-50-2
包装与价格:
包装价格(元)
2 mg电议
5 mg电议
10 mg电议
25 mg电议
50 mg电议
100 mg电议
200 mg电议
1 mL*10 mM(in DMSO)电议

产品名称
盐酸CGP71683
CGP71683A
产品介绍
CGP71683 hydrochloride 是竞争性的神经肽受体拮抗剂,Ki值为 1.3 nM。

产品描述

CGP71683 is a competitive neuropeptide Y5 receptor antagonist (Ki: 1.3 nM) and shows no obvious activity at Y1 receptor (Ki >4000 nM) and Y2 receptor (Ki: 200 nM) in cell membranes.

体内活性

CGP71683 (1-10 mg/kg, i.p.) dose-dependently decreased nocturnal and fasting-induced food intake. CGP71683A did not have an anxiogenic-like effect in the rat social interaction test. In the open-field test, carried out immediately after the elevated plus-maze test, CGP71683A inhibited horizontal and vertical activity [2].

Cas No.

192322-50-2

分子式

C26H30ClN5O2S

分子量

512.07

别名

盐酸CGP71683;CGP71683A

储存和溶解度

DMSO:120 mg/mL (234.34 mM)
H2O:10 mg/mL (19.53 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years