AC1-IN-1 是 1 型腺苷酸环化酶的选择性抑制剂(AC1,IC50 = 0.54 μM)。
产品描述
AC1-IN-1 is a selective inhibitor of adenylyl cyclase type 1 (AC1, IC50 = 0.54 μM).
体外活性
In HEK293 cells, AC1-IN-1 (30 μM, 1 hours) shows nontoxic to this human cell line[1].
体内活性
AC1-IN-1 (5.6 mg/kg; i.v.) displays modest, yet statistically significant, antiallodynic effects at 1 h post-treatment compared to the 0 min time point[1].
Cas No.
2762422-55-7
分子式
C18H18FN5O2
分子量
355.37
储存和溶解度
(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years