ADRA1D receptor agonist 1 (compound (R)-9S) is a highly potent, specific and orally bioavailable α1D adrenoceptor antagonist, with a Ki of 1.6 nM. References: [1]. Sakauchi N, et al. Discovery of 5-Chloro-1-(5-chloro-2-(methylsulfonyl)benzyl)-2-imino-1,2-dihydropyridine-3-carboxamide (TAK-259) as a Novel, Selective, and Orally Active α1D Adrenoceptor Antagonist with Antiurinary Frequency Effects: Reducing Human Ether-a-go-go-Related Gene (hERG) Liabilities. J Med Chem. 2016 Apr 14;59(7):2989-3002.

纯度：≥98%

CAS：1191908-14-1