Mutant IDH1-IN-2是突变型异柠檬酸脱氢酶蛋白抑制剂, 在荧光生物化学检测中IC50为16.6 nM，LS-MS生物化学检测中IC50为＜22 nM,。

Mutant IDH1-IN-2 is a inhibitor of mutant Isocitrate dehydrogenase (IDH) proteins, with IC50 of 16.6 nM in Fluorescence biochemical assay, IC50 of ＜22 nM in LS-MS biochemical assay.

1429176-69-1

C24H31F2N5O2

459.53

H2O:< 0.1 mg/mL (insoluble)
DMSO:50 mg/mL (108.81 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years