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GRK2-IN-1 hydrochloride(2055990-90-2 free base)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
GRK2-IN-1 hydrochloride(2055990-90-2 free base)图片
包装与价格:
包装价格(元)
1 mg电议
2 mg电议
5 mg电议
10 mg电议
25 mg电议
50 mg电议
100 mg电议
200 mg电议
500 mg电议
1 mL*10 mM(in DMSO)电议

产品名称
GRK2-IN-1 hydrochloride
产品介绍

产品描述

GRKs-IN-1 hydrochloride has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM).

体外活性

GRKs-IN-1 hydrochloride (Compound 14as) is a derivative 14as of paroxetine, shows a 100-fold improvement in cardiomyocyte contractility assays over paroxetine.

Cas No.

T13714L

分子式

C24H26ClFN4O4

分子量

488.94

别名

GRK2-IN-1 hydrochloride

储存和溶解度

DMSO:250 mg/mL (511.31 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years