CAS NO: | 30914-89-7 |
包装: | 50mg, 100mg, 250mg |
规格: | ≥98% |
Flumexadol is an orally bioavailable non-narcotic analgesic. Flumexadol is a specific and affinity 5-HT2C receptor agonist with a Ki of 25 nM for the (+)-enantiomer of Flumexadol, and is 40-fold specific over the 5-HT2A receptor. References: [1]. Hache J, et al. The pharmacology of 1841 CERM, a new analgesic. Arzneimittelforschung. 1978;28(4):642-5.
[2]. Nilsson BM. 5-Hydroxytryptamine 2C (5-HT2C) receptor agonists as potential antiobesity agents. J Med Chem. 2006 Jul 13;49(14):4023-34.
[3]. Kucharczyk N, et al. Metabolites of 2-(3-trifluoromethylphenyl)tetrahydro-1,4-oxazine (CERM) 1841) in rats and dogs. Xenobiotica. 1979 Nov;9(11):703-11.
纯度:≥98%
CAS:30914-89-7