CAY10471 Racemate 是一种高选择性的 CRTH2/DP 2 受体拮抗剂，对 hCRTH2 的Ki值为 0.6 nM，对其选择性远高于人血栓素 A2 受体 TP 或 PGD2 受体 DP。它对大小鼠的同源 CRTH2 也具有拮抗作用。

CAY 10471 is a potent, highly selective CRTH2/DP 2 receptor antagonist. CAY10471 binds to the human CRTH2/DP2, DP1, and TP receptors( Ki values of 0.6, 1200, and >10,000 nM,respectively)

844639-57-2

C21H21FN2O4S

416.47

TM30089 Racemate;3-[[(4-氟苯基)磺酰基]甲基氨基]-1,2,3,4-四氢-9H-咔唑-9-乙酸

DMSO:150 mg/mL (360.17 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years