Metergoline 是多巴胺激动剂和血清素拮抗剂。它是 h5-HT7受体的高亲和力配体,Ki为 16 nM。它还是可逆神经 Na+通道抑制剂,用于研究季节性情绪障碍、催乳激素调节。
产品描述
Metergoline is a dopamine agonist and serotonin antagonist. It has been used similarly to BROMOCRIPTINE as a dopamine agonist and also for migraine disorder therapy.
Cas No.
17692-51-2
分子式
C25H29N3O2
分子量
403.52
别名
Liserdol;甲麦角林;Methergoline
储存和溶解度
DMSO:40.4 mg/mL(100 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years