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Odapipam
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Odapipam图片
CAS NO:131796-63-9
包装:5 mg
市场价:7014元

产品名称
NNC 756
产品介绍

产品描述

Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).

体内活性

The metabolism of Odapipam has been studied with phenobarbital-induced rat liver microsomes. During the incubation of Odapipam, five different metabolites are formed. The electron-ionization (EI+) mass spectra of the metabolites indicated the formation of N-desmethyl-Odapipam, 1-hydroxy-Odapipam, the two isomers of 3′-hydroxy-Odapipam and a metabolite which is dehydrogenated in the dihydrobenzofuran moiety[1].

Cas No.

131796-63-9

分子式

C19H20ClNO2

分子量

329.82

别名

NNC 756

储存和溶解度

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years