CGP52432 是一种GABAB受体拮抗剂，IC50值为 85 nM。

CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).

Reactions are set up with Acetyl coenzyme A (AcCoA)(0.4 μM), N-terminal histone H4 peptide (sequence SGRGKGGKGLGKGGAKRHRKV-GGK-biotin)(50 nM), MOZ enzyme(10 nM), and an acetyl-lysine specific antibody (final dilution 1: 10000).

139667-74-6

C15H24Cl2NO4P

384.23

CGP 52432;4-苄氧基苯基异硫氰酸酯

DMSO:5 mg/mL (13.01 mM),Need ultrasonic and warming
Powder: -20°C for 3 years
In solvent: -80°C for 2 years