Emamectin BenzOATe 是口服有效的神经系统毒物,其通过结合昆虫中的GABA受体发挥作用。它是阿维菌素的半合成衍生物之一,具有广谱的杀虫和杀螨活性。它诱导ROS介导的 DNA 损伤和细胞凋亡。
产品描述
Emamectin Benzoate, by binding gamma-aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropods, acts as a chloride channel activator.
体外活性
Emamectin Benzoate stimulates the release of GABA from the synapses between nerve cells. It also additionally increasing GABA's affinity for its receptor on the post-junction membrane of muscle cells in insects and arthropods.
Cas No.
155569-91-8
分子式
C56H81NO15
分子量
1008.256
别名
甲胺基阿维菌素苯甲酸盐;MK-244
储存和溶解度
DMSO:31 mg/mL (16.49 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years