产品描述
GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.
体内活性
GR79236 has been shown to have antinociceptive and anti-inflammatory properties in animal models. GR79236 inhibits the release of CGRP evoked by superior sagittal sinus (SSS) stimulation in the cat and inhibits trigeminal nucleus firing in the cat and rat. GR79236X has acute, short-term analgesic efficacy.
Cas No.
124555-18-6
分子式
C15H21N5O5
分子量
351.36
别名
GR 79236
储存和溶解度
H2O:98 mg/mL (278.92 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years