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WM-3835
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
WM-3835图片
CAS NO:2229025-70-9
包装与价格:
包装价格(元)
2 mg电议
5 mg电议
10 mg电议
25 mg电议
50 mg电议
100 mg电议
200 mg电议
1 mL*10 mM(in DMSO)电议

产品介绍
WM-3835 是一种高特异性HBO1(KAT7orMYST2) 抑制剂,可直接与 HBO1 33 的乙酰辅酶 A 结合位点结合 WM-3835 激活细胞凋亡,抑制骨肉瘤细胞的增殖,迁移和侵袭。它抑制小鼠中骨肉瘤异种移植物的生长,有抗肿瘤活性。

产品描述

WM-3835 is a novel and high-specific small molecule inhibitor of Lysine Acetyltransferase 7 (KAT7, MYST2, HBO1) , able to potently suppressed OS cell proliferation and migration, and leads to apoptosis activation.

体外活性

WM-3835, a novel and high-specific small molecule HBO1 inhibitor, was able to potently suppressed OS cell proliferation and migration, and led to apoptosis activation.

Cas No.

2229025-70-9

分子式

C20H17FN2O4S

分子量

400.42

储存和溶解度

DMSO:250 mg/mL (624.34 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years