PROTAC BRD4 Degrader-1 is an efficacious degrader of BRD4(BRD4 BD1,IC50 of 41.8 nM).

PROTAC BRD4 Degrader-1 shows high inhibitory activity against the growth of human monocyte lymphoma cell line THP-1(IC50 value of 0.81 μM), and moderate activity against Raji and HL-60 cell lines[1]

2133360-00-4

C40H37N9O8

771.78

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years