[11C]MP 10 是一种特异性且有效的 PDE10A 抑制剂 (IC50=0.37 nM),其特异性活性是 PDE 的 1000 倍以上。
产品描述
[11C]MP 10, a specific and effective PDE10A inhibitor (IC50=0.37 nM), is with more than1000-fold specificity activity over the PDE.
体外活性
PF-2545920 shows excellent potency and specificity in PDE10A with IC50 of 1.26 nM.
Cas No.
1292799-56-4
别名
PF-2545920;Mardepodect
储存和溶解度
Ethanol:69 mg/mL(175.8 mM)
DMSO:79 mg/mL (201.29 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years