Tasosartan 是长效血管紧张素 II 受体拮抗剂。

Tasosartan is an antagonist of angiotensin II type 2 (AT2) receptor (IC50 = 1.2 nM).

In vivo, tasosartan (p.o. or i.v.) blocked by 80% AT1 receptors 1 to 2 h after drug administration and still had a 40% effect at 32 h.

145733-36-4

C23H21N7O

411.469

WAY-ANA 756;他索沙坦

DMSO:125 mg/mL (303.80 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years